B-Raf IN 2

CAS No. 2649372-20-1

B-Raf IN 2( —— )

Catalog No. M35194 CAS No. 2649372-20-1

B-Raf IN 2, compound Ia, is a highly effective and specific inhibitor of BRAF. It exhibits significant potential for cancer research.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 79 Get Quote
5MG 121 Get Quote
10MG 188 Get Quote
25MG 325 Get Quote
50MG 455 Get Quote
100MG 626 Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    B-Raf IN 2
  • Note
    Research use only, not for human use.
  • Brief Description
    B-Raf IN 2, compound Ia, is a highly effective and specific inhibitor of BRAF. It exhibits significant potential for cancer research.
  • Description
    B-Raf IN 2 is a potent and selective BRAF inhibitor extracted from patent WO2021116055A1, compound Ia. B-Raf IN 2 can be used for the research of cancer.
  • In Vitro
    B-Raf IN 2 shows considerably less paradoxial activation of the MAPK signaling pathway while retaining high potency.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    MAPK/ERK Signaling
  • Target
    Raf
  • Recptor
    Raf
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2649372-20-1
  • Formula Weight
    461.44
  • Molecular Formula
    C20H17F2N5O4S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (216.71 mM; Ultrasonic )
  • SMILES
    Cn1cnc2ccc(Oc3c(F)ccc(NS(=O)(=O)N4CC[C@@H](F)C4)c3C#N)cc2c1=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Dolente C, et, al. New methylquinazolinone derivatives. WO2021116055A1.
molnova catalog
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